chemical inhibits protein has role has role bromodomain-containing protein 4 inhibitor primary carboxamide pelabresib Wikipedia:CPI-0610 chebi_ontology InChI=1S/C20H16ClN3O2/c1-11-18-14-4-2-3-5-15(14)19(12-6-8-13(21)9-7-12)23-16(10-17(22)25)20(18)26-24-11/h2-9,16H,10H2,1H3,(H2,22,25)/t16-/m0/s1 Chemspider:32738784 PMID:33925695 0 Reference: PMID: 26815195 CPI0610 GCWIQUVXWZWCLE-INIZCTEOSA-N PMID:32927276 2-((4S)-6-(4-chlorophenyl)-1-methyl-4H-isoxazolo[5,4-d][2]benzazepin-4-yl)acetamide C20H16ClN3O2 CAS:1380087-89-7 PMID:26815195 CPI-0610 anhydrous CPI 0610 CPI-0610 2-[(4S)-6-(4-chlorophenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]acetamide CHEBI:189653 PMID:35114569 pelabresibum PMID:30529073 CPI-232 365.09310 PMID:31729905 An organic heterotricyclic compound that is 4H-[1,2]oxazolo[5,4-d][2]benzazepine substituted by methyl, 2-amino-2-oxoethyl, and 4-chlorophenyl groups at positions 1, 4S and 6, respectively. It is a small molecule inhibitor of bromodomain and extra-terminal (BET) proteins and exhibits antineoplastic activity. CC1=NOC2=C1C1=C(C=CC=C1)C(=NC2CC(N)=O)C1=CC=C(Cl)C=C1 PMID:32245330 PMID:33574760 365.820 PMID:27890933 PMID:33509905 pelabresib organic heterotricyclic compound inhibitor antineoplastic agent monochlorobenzenes bromodomain-containing protein 2 bromodomain-containing protein 4